Diatretol, an α, α′-dioxo-diketopiperazine, is a potent in vitro and in vivo antimalarial
Aki Ishiyama, Rei Hokari, Kenichi Nonaka, Takuya Chiba, Hiromi Miura, Kazuhiko Otoguro, Masato Iwatsuki
Topics & Concepts
In vivoPlasmodium falciparumPlasmodium bergheiIn vitroAntiparasiticMetabolitePharmacologyIC50ChemistryAntiparasitic agentBiologyMalariaBiochemistryMedicineImmunologyBiotechnologyPathologyResearch on Leishmaniasis StudiesCancer therapeutics and mechanismsQuinazolinone synthesis and applications