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Diatretol, an α, α′-dioxo-diketopiperazine, is a potent in vitro and in vivo antimalarial

Aki Ishiyama, Rei Hokari, Kenichi Nonaka, Takuya Chiba, Hiromi Miura, Kazuhiko Otoguro, Masato Iwatsuki

2021The Journal of Antibiotics17 citationsDOIOpen Access PDF

Topics & Concepts

In vivoPlasmodium falciparumPlasmodium bergheiIn vitroAntiparasiticMetabolitePharmacologyIC50ChemistryAntiparasitic agentBiologyMalariaBiochemistryMedicineImmunologyBiotechnologyPathologyResearch on Leishmaniasis StudiesCancer therapeutics and mechanismsQuinazolinone synthesis and applications
Diatretol, an α, α′-dioxo-diketopiperazine, is a potent in vitro and in vivo antimalarial | Litcius