Multifunctional quinoxaline-hydrazone derivatives with acetylcholinesterase and monoamine oxidases inhibitory activities as potential agents against Alzheimer’s disease
Ulviye Acar Çevik, Derya Osmani̇ye, Begüm Nurpelin Sağlık, Betül Kaya Çavuşoğlu, Serkan Levent, Abdullah Burak Karaduman, Sinem Ilgın, Ahmet Çağrı Karaburun, Yusuf Özkay, Zafer Asım Kaplancıklı, Gülhan Turan
Topics & Concepts
AcetylcholinesteraseButyrylcholinesteraseChemistryMonoamine oxidaseAchéQuinoxalineInhibitory postsynaptic potentialIC50Monoamine oxidase BCholinesteraseMonoamine neurotransmitterPharmacologyEnzymeIn vitroStereochemistryHydrazoneBiochemistryReceptorOrganic chemistryBiologyNeuroscienceSerotoninCholinesterase and Neurodegenerative DiseasesNicotinic Acetylcholine Receptors StudyComputational Drug Discovery Methods