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Targeted protein degradation in drug development: Recent advances and future challenges

Jian H. Song, Mingzheng Hu, Jun Zhou, Songbo Xie, Tianliang Li, Yan Li

2023European Journal of Medicinal Chemistry49 citationsDOI

Topics & Concepts

Protein degradationProteasomeChemistryDrug discoveryAutophagyUbiquitinLysosomeComputational biologyDrugDrug developmentFunction (biology)Cell biologyPharmacologyBiochemistryBiologyEnzymeGeneApoptosisProtein Degradation and InhibitorsUbiquitin and proteasome pathwaysHistone Deacetylase Inhibitors Research
Targeted protein degradation in drug development: Recent advances and future challenges | Litcius