Design, synthesis and biological evaluation of novel pleuromutilin derivatives containing piperazine and 1,2,3-triazole linker
Guang‐Yu Zhang, Zhe Zhang, Kang Li, Jie Liu, Bo Li, Zhen Jin, Yahong Liu, You‐Zhi Tang
Topics & Concepts
ChemistryPiperazineTiamulinAntibacterial activityMinimum inhibitory concentrationClick chemistryIn vivoTriazoleStaphylococcus aureusCarbohydrazideNuclear chemistryIn vitroStereochemistryAntimicrobialOrganic chemistryBiochemistryBacteriaBiologyGeneticsBiotechnologyVeterinary medicine and infectious diseasesSynthesis and Biological EvaluationQuinazolinone synthesis and applications