Litcius/Paper detail

Novel inhibitors targeting the PGK1 metabolic enzyme in glycolysis exhibit effective antitumor activity against kidney renal clear cell carcinoma in vitro and in vivo

Yu He, Yinheng Luo, Lan Huang, Dan Zhang, Huijin Hou, Yue Liang, Shi Deng, Peng Zhang, Shufang Liang

2024European Journal of Medicinal Chemistry18 citationsDOIOpen Access PDF

Topics & Concepts

GlycolysisChemistryIn vivoEnzymeSorafenibCell growthBiochemistryMetabolic pathwayKidneyCancer researchPharmacologyBiologyEndocrinologyHepatocellular carcinomaBiotechnologyRenal cell carcinoma treatmentEpigenetics and DNA MethylationCancer, Hypoxia, and Metabolism