Discovery of novel flavonoid derivatives as potential dual inhibitors against α-glucosidase and α-amylase: virtual screening, synthesis, and biological evaluation
Tan Thanh, Minh-Hoang Phan, Thao Thi Thai, Thua-Phong Lam, Nghia Vo-Trong Lai, Thanh-Thao Nguyen, Thuy-Viet-Phuong Nguyen, Cam‐Van T. Vo, Khac‐Minh Thai, Thanh‐Dao Tran
Topics & Concepts
AcarboseFlavonoidEnzymeVirtual screeningIC50ChemistryDiabetes mellitusAmylaseDocking (animal)PharmacologyIn vitroBiochemistryMedicineDrug discoveryAntioxidantNursingEndocrinologyNatural Antidiabetic Agents StudiesEnzyme Production and CharacterizationDiet, Metabolism, and Disease