Lipase-catalysed one-pot synthesis of thiazole-based Betti bases and their evaluation as potential cholinesterase inhibitors
Sarfaraz Shaikh, M. M. V. Ramana
Topics & Concepts
ChemistryThiazoleLipaseCholinesteraseAcetylcholinesteraseIC50ButyrylcholinesteraseAchéStereochemistryGalantamineIn vitroEnzymeBiochemistryPharmacologyBiologyDiseaseDonepezilMedicinePathologyDementiaCholinesterase and Neurodegenerative DiseasesComputational Drug Discovery MethodsChemical synthesis and alkaloids