Crystal structure of human acetylcholinesterase in complex with tacrine: Implications for drug discovery
K.V. Dileep, Kentaro Ihara, Chiemi Mishima-Tsumagari, Mutsuko Kukimoto‐Niino, Mayumi Yonemochi, Kazuharu Hanada, Mikako Shirouzu, Kam Y. J. Zhang
Topics & Concepts
TacrineAcetylcholinesteraseCholinergicChemistryAcetylcholineDrug discoveryDrugPharmacologyAchéAcetylcholinesterase inhibitorNeuroscienceBiophysicsBiochemistryPsychologyMedicineBiologyEnzymeCholinesterase and Neurodegenerative DiseasesComputational Drug Discovery MethodsChemical synthesis and alkaloids