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Crystal structure of human acetylcholinesterase in complex with tacrine: Implications for drug discovery

K.V. Dileep, Kentaro Ihara, Chiemi Mishima-Tsumagari, Mutsuko Kukimoto‐Niino, Mayumi Yonemochi, Kazuharu Hanada, Mikako Shirouzu, Kam Y. J. Zhang

2022International Journal of Biological Macromolecules144 citationsDOI

Topics & Concepts

TacrineAcetylcholinesteraseCholinergicChemistryAcetylcholineDrug discoveryDrugPharmacologyAchéAcetylcholinesterase inhibitorNeuroscienceBiophysicsBiochemistryPsychologyMedicineBiologyEnzymeCholinesterase and Neurodegenerative DiseasesComputational Drug Discovery MethodsChemical synthesis and alkaloids
Crystal structure of human acetylcholinesterase in complex with tacrine: Implications for drug discovery | Litcius