Synthesis, biological evaluation and docking studies of silicon incorporated diarylpyrroles as MmpL3 inhibitors: An effective strategy towards development of potent anti-tubercular agents
N. Vasudevan, Zenia Motiwala, Remya Ramesh, Sachin Bhausaheb Wagh, Rahul D. Shingare, Revansiddha Katte, Amitesh Anand, Sushil Choudhary, Ajay Kumar, Rajesh S. Gokhale, Kiran Kulkarni, D. Srinivasa Reddy
Topics & Concepts
ChemistryPharmacophoreDocking (animal)Mycobacterium tuberculosisADMEMycolic acidResazurinStereochemistryVirtual screeningCombinatorial chemistryLead compoundBiochemistryDrug discoveryIn vitroTuberculosisPathologyNursingMedicineTuberculosis Research and EpidemiologyCancer therapeutics and mechanismsPneumocystis jirovecii pneumonia detection and treatment