Discovery of BP3 as an efficacious proteolysis targeting chimera (PROTAC) degrader of HSP90 for treating breast cancer
Quanyu Liu, Guihui Tu, Yan Hu, Qingna Jiang, Jingwen Liu, Shanshan Lin, Zelei Yu, Ge Li, Xinhua Wu, Yuanling Tang, Xiuwang Huang, Jianhua Xu, Yang Liu, Lixian Wu
Topics & Concepts
Hsp90ProteolysisChemistryChimera (genetics)CancerBreast cancerHeat shock proteinHsp90 inhibitorCancer researchPharmacologyBiochemistryMedicineEnzymeInternal medicineGeneUbiquitin and proteasome pathwaysPeptidase Inhibition and AnalysisProtein Degradation and Inhibitors