Litcius/Paper detail

Novel hydroxybenzylamine-deoxyvasicinone hybrids as anticholinesterase therapeutics for Alzheimer’s disease

Suresh K. Bowroju, Narsimha Reddy Penthala, Naga Rajiv Lakkaniga, Meenakshisundaram Balasubramaniam, Srinivas Ayyadevara, Robert J. Shmookler Reis, Peter A. Crooks

2021Bioorganic & Medicinal Chemistry22 citationsDOIOpen Access PDF

Topics & Concepts

ButyrylcholinesteraseChemistryAcetylcholinesteraseAllosteric regulationAchéPeptideIC50EnzymeStereochemistryBiochemistryIn vitroCholinesterase and Neurodegenerative DiseasesComputational Drug Discovery MethodsNicotinic Acetylcholine Receptors Study