Novel hydroxybenzylamine-deoxyvasicinone hybrids as anticholinesterase therapeutics for Alzheimer’s disease
Suresh K. Bowroju, Narsimha Reddy Penthala, Naga Rajiv Lakkaniga, Meenakshisundaram Balasubramaniam, Srinivas Ayyadevara, Robert J. Shmookler Reis, Peter A. Crooks
Topics & Concepts
ButyrylcholinesteraseChemistryAcetylcholinesteraseAllosteric regulationAchéPeptideIC50EnzymeStereochemistryBiochemistryIn vitroCholinesterase and Neurodegenerative DiseasesComputational Drug Discovery MethodsNicotinic Acetylcholine Receptors Study