Cryo-EM Structure of K+-Bound hERG Channel Complexed with the Blocker Astemizole
Tatsuki Asai, Naruhiko Adachi, Toshio Moriya, Hideyuki Oki, Takamitsu Maru, Masato Kawasaki, K. Suzuki, Si-Si Chen, Ryohei Ishii, Kazuko Yonemori, S. Igaki, Satoshi Yasuda, Satoshi Ogasawara, Toshiya Senda, Takeshi Murata
Topics & Concepts
hERGAstemizolePotassium channelPotassium channel blockerChemistryPharmacologyBiophysicsRepolarizationElectrophysiologyInternal medicineMedicineBiologyForce Microscopy Techniques and ApplicationsCardiac electrophysiology and arrhythmiasIntegrated Circuits and Semiconductor Failure Analysis