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Synthesis and anti-MRSA activity of quaternized small molecule antimicrobial peptide mimics based on norharmane

Wenjia Dan, Yingyan Xiong, Runchu Li, Hui Gao, Panpan Liu, Meixia Sui, Chenggong Xu, Jiangkun Dai

2025European Journal of Medicinal Chemistry12 citationsDOI

Topics & Concepts

ChemistryAntimicrobialPeptideCombinatorial chemistryMoleculeSmall moleculeStereochemistryAntibacterial agentAntibioticsOrganic chemistryBiochemistrySynthesis and bioactivity of alkaloidsBioactive Compounds and Antitumor AgentsCancer therapeutics and mechanisms
Synthesis and anti-MRSA activity of quaternized small molecule antimicrobial peptide mimics based on norharmane | Litcius