The novel dual-mechanism Kv7 potassium channel/TSPO receptor activator GRT-X is more effective than the Kv7 channel opener retigabine in the 6-Hz refractory seizure mouse model
Petra Bloms‐Funke, Marion Bankstahl, Jens P. Bankstahl, Christa Kneip, Wolfgang Schröder, Wolfgang Löscher
Topics & Concepts
PharmacologyEpilepsyPotassium channelNeuroprotectionChemistryNeuroactive steroidTranslocator proteinAllosteric regulationAnxiolyticAnticonvulsantSeizure thresholdMedicineNeurosciencePsychologyInternal medicineReceptorGABAA receptorInflammationNeuroinflammationIon channel regulation and functionNeuroscience and Neuropharmacology ResearchCardiac electrophysiology and arrhythmias