Litcius/Paper detail

PTMs as molecular encoders: reprogramming chaperones into epichaperomes for network control in disease

Feixia Chu, Sahil Sharma, Stephen D. Ginsberg, Gabriela Chiosis

2025Trends in Biochemical Sciences9 citationsDOIOpen Access PDF

Abstract

Recent discoveries reveal that post-translational modifications (PTMs) do more than regulate protein activity - they encode conformational states that transform chaperones into epichaperomes: multimeric scaffolds that rewire protein-protein interaction networks. This emerging paradigm expands the framework of chaperone biology in disease and provides a structural basis for systems-level dysfunction in disorders such as cancer and Alzheimer's disease. This review explores how PTMs within intrinsically disordered regions drive epichaperome formation, how these scaffolds selectively regulate disease-enabling functions, and why their disruption normalizes pathological networks. By highlighting PTMs as molecular encoders of supramolecular assemblies, we propose a shift from targeting proteins to targeting network architectures that sustain and perpetuate disease - a concept with broad implications for cell biology, disease propagation, and therapeutic design.

Topics & Concepts

ReprogrammingComputational biologyDiseaseEncoderControl (management)BiologyComputer scienceCell biologyChemistryGeneticsMedicineArtificial intelligenceGeneInternal medicineOperating systemRNA modifications and cancerRNA Research and SplicingCancer-related molecular mechanisms research