Hyperactivation of TORC1 Drives Resistance to the Pan-HER Tyrosine Kinase Inhibitor Neratinib in HER2-Mutant Cancers
Dhivya R. Sudhan, Ángel Guerrero‐Zotano, Helen Won, Paula González Ericsson, Alberto Servetto, Mariela Huerta-Rosario, Dan Ye, Kyung‐min Lee, Luigi Formisano, Yan Guo, Qi Liu, Lisa N. Kinch, Monica Red Brewer, Teresa C. Dugger, James P. Koch, Michael J. Wick, Richard E. Cutler, Alshad S. Lalani, Richard Bryce, Alan Auerbach, Ariella B. Hanker, Carlos L. Arteaga
Topics & Concepts
NeratinibLapatinibCancer researchTyrosine-kinase inhibitorEndocytic cycleTyrosine kinaseCell biologyChemistryBiologyEndocytosisCancerSignal transductionCellGeneticsBreast cancerTrastuzumabHER2/EGFR in Cancer Research