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Carboxylesterase Notum Is a Druggable Target to Modulate Wnt Signaling

Elliott D. Bayle, Fredrik Svensson, Benjamin N. Atkinson, David Steadman, Nicky J. Willis, Hannah L. Woodward, Paul J. Whiting, Jean‐Paul Vincent, Paul V. Fish

2021Journal of Medicinal Chemistry49 citationsDOIOpen Access PDF

Abstract

), which are complementary chemical tools for exploring the role of Notum in Wnt signaling.

Topics & Concepts

Wnt signaling pathwayDruggabilityComputational biologyRegulatorSignal transductionBiologyCell biologyGeneticsGeneWnt/β-catenin signaling in development and cancerCholinesterase and Neurodegenerative DiseasesCancer-related gene regulation
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