In vitro and in silico inhibitory effects of synthetic and natural eugenol derivatives against the NorA efflux pump in Staphylococcus aureus
Débora Feitosa Muniz, Cristina Rodrigues dos Santos Barbosa, Irwin Rose Alencar de Menezes, Erlânio Oliveira de Sousa, Raimundo Luíz Silva Pereira, João Tavares Calixto Júnior, Pedro Silvino Pereira, Yedda Maria Lobo Soares de Matos, Roger Henrique Sousa da Costa, Cícera Datiane de Morais Oliveira–Tintino, Henrique Douglas Melo Coutinho, José Maria Barbosa‐Filho, Gabriela Ribeiro de Sousa, Jaime Ribeiro‐Filho, José P. Siqueira-Júnior, Saulo Relison Tintino
Topics & Concepts
Ethidium bromideEugenolEffluxChemistryIsoeugenolNorfloxacinAntibacterial activityStaphylococcus aureusMinimum inhibitory concentrationBiochemistryIn vitroAntibioticsBacteriaOrganic chemistryBiologyCiprofloxacinGeneticsDNAPhenothiazines and Benzothiazines Synthesis and ActivitiesAntimicrobial Resistance in StaphylococcusAntibiotics Pharmacokinetics and Efficacy