Discovery of novel VEGFR-2 inhibitors embedding 6,7-dimethoxyquinazoline and diarylamide fragments
Ru Wang, Hu Liu, Yuanyuan You, Xinyu Wang, Bingbing Lv, Liqin Cao, Jia‐Yu Xue, Yungen Xu, Lei Shi
Topics & Concepts
ChemistryDocking (animal)VEGF receptorsIn vitroStereochemistryMoietyStructure–activity relationshipIC50AngiogenesisKinaseCell cultureBiochemistryCancer researchMedicineBiologyNursingGeneticsAngiogenesis and VEGF in CancerHER2/EGFR in Cancer ResearchQuinazolinone synthesis and applications