Kinetic and structural studies on the inhibition of acetylcholinesterase and butyrylcholinesterase by a series of multitarget-directed galantamine-peptide derivatives
Alessandro Pesaresi, Doriano Lamba, L. Vezenkov, Daniela S. Tsekova, Valentin Lozanov
Topics & Concepts
ButyrylcholinesteraseGalantamineAcetylcholinesterasePharmacologyChemistryCholinesteraseDocking (animal)PeptideAnticholinergicAcetylcholinesterase inhibitorEnzymeDonepezilBiochemistryMedicineAchéDiseaseDementiaInternal medicineNursingCholinesterase and Neurodegenerative DiseasesComputational Drug Discovery MethodsChemical synthesis and alkaloids