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CHI3L1-targeted small molecules as glioblastoma therapies: Virtual screening-based discovery, biophysical validation, pharmacokinetic profiling, and evaluation in glioblastoma spheroids

Hossam Nada, Longfei Zhang, Baljit Kaur, Moustafa T. Gabr

2025European Journal of Medicinal Chemistry18 citationsDOIOpen Access PDF

Topics & Concepts

GlioblastomaChemistrySpheroidSmall moleculeProfiling (computer programming)PharmacokineticsVirtual screeningDrug discoveryPharmacologyComputational biologyCancer researchIn vitroMedicineBiologyBiochemistryOperating systemComputer scienceStudies on Chitinases and ChitosanasesAdvanced biosensing and bioanalysis techniquesRNA Interference and Gene Delivery
CHI3L1-targeted small molecules as glioblastoma therapies: Virtual screening-based discovery, biophysical validation, pharmacokinetic profiling, and evaluation in glioblastoma spheroids | Litcius