Litcius/Paper detail

Novel 4-aminoquinolines: Synthesis, inhibition of the Mycobacterium tuberculosis enoyl-acyl carrier protein reductase, antitubercular activity, SAR, and preclinical evaluation

Josiane Delgado Paz, Nathalia Sperotto, Alessandro Silva Ramos, Kenia Pissinate, Valnês S. Rodrigues-Junior, Bruno Lopes Abbadi, Ana Flávia Borsoi, Raoní Scheibler Rambo, Ana Carolina Corso Minotto, Adílio da Silva Dadda, Luiza Galina, Fernanda Souza Macchi Hopf, Mauro Neves Muniz, Leonardo Martinelli, Candida Deves Roth, Rodrigo Braccini Madeira Silva, Marcia Alberton Perelló, Alexia de Matos Czeczot, Christiano Ev Neves, Lovaine Silva Duarte, Mariana Leyser, Sı́lvia Dias de Oliveira, Cristiano Valim Bizarro, Pablo Machado, Luiz Augusto Basso

2022European Journal of Medicinal Chemistry19 citationsDOIOpen Access PDF

Topics & Concepts

Mycobacterium tuberculosisChemistryADMEIn vivoPharmacologyVirtual screeningIn vitroTuberculosisReductaseToxicityEnzymeBiochemistryDrug discoveryBiologyMedicineBiotechnologyOrganic chemistryPathologyTuberculosis Research and EpidemiologyAntibiotic Resistance in BacteriaPneumocystis jirovecii pneumonia detection and treatment