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Stereospecific Isomerization of Allylic Halides via Ion Pairs with Induced Noncovalent Chirality

Samuel Martinez‐Erro, Víctor García‐Vázquez, Amparo Sanz‐Marco, Belén Martín‐Matute

2020Organic Letters23 citationsDOIOpen Access PDF

Abstract

ratios. Furthermore, the [1,3]-proton shift takes place with an outstanding level of chirality transfer from chiral allylic alcohols (≤98%) to give chiral trifluoromethylated vinyl chlorides.

Topics & Concepts

Allylic rearrangementChemistryChirality (physics)IsomerizationStereospecificityHalideRegioselectivityEnantioselective synthesisCatalysisProtonMedicinal chemistryOrganic chemistryPhysicsQuantum mechanicsChiral symmetry breakingQuarkNambu–Jona-Lasinio modelFluorine in Organic ChemistryAsymmetric Synthesis and CatalysisChemical Synthesis and Analysis
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