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Crystal structure of O-Acetylserine sulfhydralase (OASS) isoform 3 from Entamoeba histolytica: Pharmacophore-based virtual screening and validation of novel inhibitors

Sudhaker Dharavath, Ramachandran Vijayan, Khushboo Kumari, Priya Tomar, Samudrala Gourinath

2020European Journal of Medicinal Chemistry18 citationsDOI

Topics & Concepts

Entamoeba histolyticaChemistryPharmacophoreGene isoformCysteineGene knockdownDeubiquitinating enzymeEnzymeBiochemistryStereochemistryGeneBiologyGeneticsUbiquitinBiochemical and Molecular ResearchNitrogen and Sulfur Effects on BrassicaFolate and B Vitamins Research
Crystal structure of O-Acetylserine sulfhydralase (OASS) isoform 3 from Entamoeba histolytica: Pharmacophore-based virtual screening and validation of novel inhibitors | Litcius