Development of anti-breast cancer PI3K inhibitors based on 7-azaindole derivatives through scaffold hopping: Design, synthesis and in vitro biological evaluation
Chengbin Yang, Mingzhu Lu, Yi Chen, Ruiqing Xiang, Tianze Qiu, Jia Yu, Yongtai Yang, Xiaofeng Liu, Mingli Deng, Yun Ling, Yaming Zhou
Topics & Concepts
PI3K/AKT/mTOR pathwayChemistryBreast cancerIn vitroCancerKinaseProtein kinase BCell growthApoptosisIntracellularCancer cellCancer researchPharmacologyBiochemistryBiologyInternal medicineMedicinePI3K/AKT/mTOR signaling in cancerSynthesis and biological activityProtein Degradation and Inhibitors