Litcius/Paper detail

Discovery of a series of ester-substituted NLRP3 inflammasome inhibitors

David Harrison, Nicolas Boutard, Krzysztof Brzózka, Marta Bugaj, Stefan Chmielewski, Anna Cierpich, John R. Doedens, Charles-Henry R.Y. Fabritius, Christopher A. Gabel, Michał Gałȩzowski, Piotr Kowalczyk, Oleksandr Levenets, Magdalena Mroczkowska, Katarzyna Palica, Roderick A. Porter, D. Schultz, Marta Sowińska, Grzegorz Topolnicki, Piotr Urbański, Jakub Woyciechowski, Alan P. Watt

2020Bioorganic & Medicinal Chemistry Letters30 citationsDOIOpen Access PDF

Topics & Concepts

InflammasomeChemistryProinflammatory cytokinePharmacologyEnzymeDrug discoveryDrugInflammationBiochemistryReceptorImmunologyMedicineInflammasome and immune disordersTryptophan and brain disordersAdenosine and Purinergic Signaling