Discovery of a series of ester-substituted NLRP3 inflammasome inhibitors
David Harrison, Nicolas Boutard, Krzysztof Brzózka, Marta Bugaj, Stefan Chmielewski, Anna Cierpich, John R. Doedens, Charles-Henry R.Y. Fabritius, Christopher A. Gabel, Michał Gałȩzowski, Piotr Kowalczyk, Oleksandr Levenets, Magdalena Mroczkowska, Katarzyna Palica, Roderick A. Porter, D. Schultz, Marta Sowińska, Grzegorz Topolnicki, Piotr Urbański, Jakub Woyciechowski, Alan P. Watt
Topics & Concepts
InflammasomeChemistryProinflammatory cytokinePharmacologyEnzymeDrug discoveryDrugInflammationBiochemistryReceptorImmunologyMedicineInflammasome and immune disordersTryptophan and brain disordersAdenosine and Purinergic Signaling