Novel thieno[2,3-b]quinoline-procaine hybrid molecules: A new class of allosteric SHP-1 activators evolved from PTP1B inhibitors
Lei Xu, Xu-Yang Mu, Minmin Liu, Zhijia Wang, Chao Shen, Qianwen Mu, Bo Feng, Yechun Xu, Tingjun Hou, Lixin Gao, Haini Jiang, Jia Li, Yubo Zhou, Wenlong Wang
Topics & Concepts
Allosteric regulationChemistrySmall moleculeSignal transductionIn vitroBiochemistryEnzymeCancer researchCell biologyBiologyProtein Tyrosine PhosphatasesCytokine Signaling Pathways and InteractionsGalectins and Cancer Biology