Thiosemicarbazone derivatives as potential inhibitors of acetylcholinesterase, butyrylcholinesterase and their molecular docking studies
Asla Abdullah AL-Zahrani, Nasser S. Awwad, Hala A. Ibrahium, Shawkat Hayat, Hayat Ullah, Zarqa Javed, Fazal Rahim, Muhammad Saleem Khan, Hussan Zada, Abdur Rab, Khalid Raza, Abdul Wadood
Topics & Concepts
ButyrylcholinesteraseAcetylcholinesteraseAchéDocking (animal)SemicarbazoneIC50CholinesteraseChemistryEnzymePharmacologyStereochemistryDrugEnzyme inhibitionBiochemistryMedicineIn vitroNursingCholinesterase and Neurodegenerative DiseasesComputational Drug Discovery MethodsSynthesis and biological activity