An overview of compound properties, multiparameter optimization, and computational drug design methods for PARP-1 inhibitor drugs
Bhakti Umesh Hirlekar, Anila Nuthi, Krishan Dev Singh, Upadhyayula Suryanarayana Murty, Vaibhav A. Dixit
Topics & Concepts
DrugRational designComputational biologyChemistryPoly ADP ribose polymerasePharmacologyAnticancer drugCombinatorial chemistryNanotechnologyMedicineBiologyBiochemistryMaterials scienceEnzymePolymerasePARP inhibition in cancer therapyComputational Drug Discovery MethodsPlant Genetic and Mutation Studies