A minimally-masked inactive prodrug of panobinostat that is bioorthogonally activated by gold chemistry
Belén Rubio‐Ruíz, Ana M. Pérez‐López, Víctor Sebastián, Asier Unciti‐Broceta
Topics & Concepts
PanobinostatProdrugChemistryBioorthogonal chemistryCombinatorial chemistryChemical synthesisIn vitroBiochemistryClick chemistryHistone deacetylaseGeneHistoneClick Chemistry and ApplicationsHistone Deacetylase Inhibitors ResearchPeptidase Inhibition and Analysis