Modulation of estrogen-related receptors subtype selectivity: Conversion of an ERRβ/γ selective agonist to ERRα/β/γ pan agonists
Mohamed G. Shahien, Mohamed Elagawany, Sadichha Sitaula, Shaimaa S. Goher, Sheryl L. Burris, Ryan Sanders, Amer Avdagic, Cyrielle Billon, Lamees Hegazy, Thomas P. Burris, Bahaa Elgendy
Topics & Concepts
ChemistryAgonistFunctional selectivityNuclear receptorReceptorEnergy homeostasisAllosteric regulationPharmacologyCell biologyBiochemistryTranscription factorGeneBiologyEstrogen and related hormone effectsReceptor Mechanisms and SignalingComputational Drug Discovery Methods