Synthesis of novel N-phenylbenzamide-thiazoles with potential DHFR inhibitory activity: Antibacterial activity, DFT and ADMET studies
Salwa Magdy Eldaly, Hamdi M. Hassaneen, Nadia Hanafy Metwally
Topics & Concepts
ChemistryAntibacterial activityCombinatorial chemistryInhibitory postsynaptic potentialStereochemistryMinimum inhibitory concentrationComputational chemistryAntimicrobialOrganic chemistryBacteriaGeneticsBiologyNeuroscienceSynthesis and biological activitySynthesis of heterocyclic compoundsSulfur-Based Synthesis Techniques