Discovery of 1,2,3-triazole incorporated indole-piperazines as potent antitubercular agents: Design, synthesis, in vitro biological evaluation, molecular docking and ADME studies
Rajkumar Reddyrajula, Umadevi Etikyala, Vijjulatha Manga, Udayakumar Dalimba
Topics & Concepts
ChemistryADMEPiperazineAntimycobacterialPyrazinamideIsoniazidIndole testMycobacterium tuberculosisDocking (animal)StereochemistryIn vitroBiochemistryAntibioticsOrganic chemistryTuberculosisRifampicinMedicinePathologyNursingTuberculosis Research and EpidemiologySynthesis and biological activityClick Chemistry and Applications