Identification and optimization of piperlongumine analogues as potential antioxidant and anti-inflammatory agents via activation of Nrf2
Limei Ji, Lailiang Qu, Cheng Wang, Wan Peng, Shang Li, Huali Yang, Heng Luo, Fucheng Yin, Dehua Lu, Xingchen Liu, Lingyi Kong, Xiaobing Wang
Topics & Concepts
GCLMOxidative stressChemistryGCLCKEAP1AntioxidantNeuroprotectionDownregulation and upregulationInflammationPharmacologySignal transductionNeurodegenerationReactive oxygen speciesBiochemistryCell biologyTranscription factorImmunologyBiologyDiseaseGeneMedicinePathologyPiperaceae Chemical and Biological StudiesCholinesterase and Neurodegenerative DiseasesMedicinal Plants and Neuroprotection