Design, synthesis and biological evaluation of novel benzofuran derivatives as potent LSD1 inhibitors
Xiangyu Zhang, Hai‐Lan Huang, Ziheng Zhang, Jiangkun Yan, Tianxiao Wu, Wenbo Yin, Yixiang Sun, Xinran Wang, Yanting Gu, Dongmei Zhao, Maosheng Cheng
Topics & Concepts
ChemistryBenzofuranChemical synthesisCombinatorial chemistryBiological activityStereochemistryBiochemistryIn vitroEpigenetics and DNA MethylationChemical Reactions and IsotopesNeuroendocrine regulation and behavior