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Site‐Selective (<i>Z</i>)‐α‐Borylalkenyl Copper Systems for Nucleophilic Stereodefined Allylic Coupling

Mireia Pujol, Ricardo J. Maza, Oriol Salvadó, Jorge J. Carbó, Elena Fernández

2022Angewandte Chemie International Edition15 citationsDOIOpen Access PDF

Abstract

Abstract 1,1‐Diborylalkenes can be transformed into ( Z )‐skipped dienes through Cu I ‐phosphine catalyzed allylic coupling reactions. The energetically preferred formation of ( Z )‐α‐borylalkenyl copper (I) species and the subsequent nucleophilic attack, explains the stereoselective nucleophilic substitution with allyl bromides. The eventual treatment of ( Z )‐skipped dienes with NaO t Bu promotes cyclization/aromatization patterns via enyne intermediates.

Topics & Concepts

Allylic rearrangementCopperNucleophileCoupling (piping)ChemistryCrystallographyStereochemistryMaterials scienceMetallurgyOrganic chemistryCatalysisOrganoboron and organosilicon chemistryCatalytic Cross-Coupling ReactionsOrganometallic Complex Synthesis and Catalysis