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Poly (ADP-ribose) polymerase (PARP) inhibitors as anticancer agents: An outlook on clinical progress, synthetic strategies, biological activity, and structure-activity relationship

Pronoy Kanti Das, Gurubasavaraja Swamy Purawarga Matada, Rohit Pal, Lalmohan Maji, Prasad Sanjay Dhiwar, B V Manjushree, Mayavan Viji

2024European Journal of Medicinal Chemistry24 citationsDOIOpen Access PDF

Topics & Concepts

Poly ADP ribose polymeraseDNA repairPolymeraseSynthetic lethalityDNA damageChemistryOlaparibPharmacologyDNACancer researchBiochemistryBiologyPARP inhibition in cancer therapyIntegrated Circuits and Semiconductor Failure AnalysisDNA Repair Mechanisms
Poly (ADP-ribose) polymerase (PARP) inhibitors as anticancer agents: An outlook on clinical progress, synthetic strategies, biological activity, and structure-activity relationship | Litcius