The emerging landscape of peptide-based inhibitors of PCSK9
Benjamin J. Tombling, Yuhui Zhang, Yen‐Hua Huang, David J. Craik, Conan K. Wang
Topics & Concepts
PCSK9Proprotein convertaseKexinPharmacologyPeptidomimeticAlirocumabMedicineMonoclonal antibodyEvolocumabDrug discoveryPotencyDrugSubtilisinPeptideAntibodyComputational biologyLDL receptorBioinformaticsBiologyCholesterolImmunologyBiochemistryApolipoprotein BInternal medicineIn vitroLipoproteinEnzymeApolipoprotein A1Lipoproteins and Cardiovascular HealthMonoclonal and Polyclonal Antibodies ResearchBiosimilars and Bioanalytical Methods