Comparison of the inhibitory effects of azole antifungals on cytochrome P450 3A4 genetic variants
Yuki Yamaguchi, Takeshi Akiyoshi, Go Kawamura, Ayuko Imaoka, Mitsue Miyazaki, F. Peter Guengerich, Katsunori Nakamura, Koujirou Yamamoto, Hisakazu Ohtani
Topics & Concepts
KetoconazoleCYP3A4ItraconazoleAzoleVoriconazoleFluconazolePharmacologyCytochrome P450ChemistryDrug interactionDrugEnzymeBiologyMicrobiologyAntifungalBiochemistryPharmacogenetics and Drug MetabolismInflammatory mediators and NSAID effectsBiosimilars and Bioanalytical Methods