Design and synthesis of new triarylimidazole derivatives as dual inhibitors of BRAFV600E/p38α with potential antiproliferative activity
Bahaa G. M. Youssif, Ahmed M. Gouda, Amr H. Moustafa, Antar A. Abdelhamid, Hesham A. M. Gomaa, Islam Kamal, Adel A. Marzouk
Topics & Concepts
ChemistryMoietyDocking (animal)StereochemistryImidazoleArylCombinatorial chemistryIn vitroOxadiazoleBiochemistryOrganic chemistryMedicineNursingAlkylMelanoma and MAPK PathwaysCytokine Signaling Pathways and InteractionsProtein Kinase Regulation and GTPase Signaling