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YB-1 Phosphorylation at Serine 209 Inhibits Its Nuclear Translocation

Ekaterina M. Sogorina, Ekaterina R. Kim, Alexey V. Sorokin, Dmitry N. Lyabin, Lev P. Ovchinnikov, Daria A. Mordovkina, Irina A. Eliseeva

2021International Journal of Molecular Sciences17 citationsDOIOpen Access PDF

Abstract

YB-1 is a multifunctional DNA- and RNA-binding protein involved in cell proliferation, differentiation, and migration. YB-1 is a predominantly cytoplasmic protein that is transported to the nucleus in certain conditions, including DNA-damaging stress, transcription inhibition, and viral infection. In tumors, YB-1 nuclear localization correlates with high aggressiveness, multidrug resistance, and a poor prognosis. It is known that posttranslational modifications can regulate the nuclear translocation of YB-1. In particular, well-studied phosphorylation at serine 102 (S102) activates YB-1 nuclear import. Here, we report that Akt kinase phosphorylates YB-1 in vitro at serine 209 (S209), which is located in the vicinity of the YB-1 nuclear localization signal. Using phosphomimetic substitutions, we showed that S209 phosphorylation inhibits YB-1 nuclear translocation and prevents p-S102-mediated YB-1 nuclear import.

Topics & Concepts

PhosphorylationNuclear transportSerineNuclear localization sequenceCell nucleusCell biologyKinaseNuclear proteinBiologyChromosomal translocationProtein kinase BCytoplasmTranscription (linguistics)Transcription factorNuclear export signalMolecular biologyChemistryBiochemistryGenePhilosophyLinguisticsRNA Research and SplicingHeat shock proteins researchRNA and protein synthesis mechanisms