Design and synthesis of certain 7-Aryl-2-Methyl-3-Substituted Pyrazolo{1,5-a}Pyrimidines as multikinase inhibitors
Mustafa A. Al-Qadhi, Heba Abdelrasheed Allam, Samar H. Fahim, Tawfeek Ahmed Ali Yahya, Fatma A.F. Ragab
Topics & Concepts
ChemistryStereochemistryIC50EnzymeDocking (animal)PharmacophoreArylCell cycle checkpointStructure–activity relationshipKinaseLead compoundApoptosisInhibitory postsynaptic potentialIn vitroCell cycleBiochemistryAlkylOrganic chemistryMedicineNeuroscienceNursingBiologyCancer Mechanisms and TherapyQuinazolinone synthesis and applicationsCancer therapeutics and mechanisms