Fragment merging approach for the design of thiazole/thiazolidine clubbed pyrazoline derivatives as anti-inflammatory agents: Synthesis, biopharmacological evaluation and molecular modeling studies
Mohamed K. Elgohary, Soha R. Abd El Hadi, Mahmoud F. Abo-Ashour, Mohammed E. Abo‐El Fetoh, Hassan Afify, Hatem A. Abdel‐Aziz, Sahar M. Abou‐Seri
Topics & Concepts
ChemistryThiazoleThiazolidinePyrazolineIn vivoCelecoxibIC50PharmacologyStereochemistryCombinatorial chemistryAnti-inflammatoryBiochemistryIn vitroMedicinal chemistryMedicineBiologyBiotechnologySynthesis and biological activitySynthesis and Biological EvaluationInflammatory mediators and NSAID effects