New TRPM8 blockers exert anticancer activity over castration-resistant prostate cancer models
Veronica Di Sarno, Pia Giovannelli, Alicia Medina-Peris, Tania Ciaglia, Marzia Di Donato, Simona Musella, Gianluigi Lauro, Vincenzo Vestuto, Gerardina Smaldone, Francesca Di Matteo, Giuseppe Bifulco, Gabriella Castoria, Antimo Migliaccio, Asia Fernández‐Carvajal, Pietro Campiglia, Isabel Gómez‐Monterrey, Carmine Ostacolo, Alessia Bertamino
Topics & Concepts
Prostate cancerChemistryDruggabilityPharmacologyTRPM8ProstateCancerBiochemistryReceptorInternal medicineMedicineGeneTransient receptor potential channelTRPV1Ion Channels and Receptors