Synthesis, antidiabetic activity and in silico studies of benzo[b]thiophene based small molecule α-amylase inhibitors
Rupal J. Joshi, Monil P. Dholariya, Savankumar R. Chothani, Chirag A. Chamakiya, Hardik L. Varu, Manisha B. Karmur, Deepika Maliwal, Raghuvir R. S. Pissurlenkar, Atul H. Bapodra, Anil S. Patel, Naval Kapuriya
Topics & Concepts
ChemistryThiopheneSmall moleculeIC50StereochemistryContext (archaeology)AmylaseIn silicoAcarboseEnzymeActive siteBiochemistryIn vitroOrganic chemistryBiologyGenePaleontologyClick Chemistry and ApplicationsNuclear Receptors and SignalingComputational Drug Discovery Methods