Combined ligand-based and structure-based design of PDE 9A inhibitors against Alzheimer’s disease
Rayala Swetha, A. Sharma, Ravi Singh, Ankit Ganeshpurkar, Devendra Kumar, Ashok Kumar, Sushil Kumar Singh
Topics & Concepts
Docking (animal)Virtual screeningChemistryPostsynaptic potentialPharmacophoreSynaptic plasticityComputational biologyLigand (biochemistry)Drug discoveryNMDA receptorNeuroscienceBiochemistryBiologyReceptorMedicineNursingCholinesterase and Neurodegenerative DiseasesComputational Drug Discovery MethodsPhosphodiesterase function and regulation