Sulfonamide-Pyrazole derivatives as next-generation Cyclooxygenase-2 enzyme inhibitors: From molecular design to in vivo efficacy
Mohamed K. Elgohary, Mahmoud S. Elkotamy, Mahmoud Abdelrahman Alkabbani, Mahmoud A. El Hassab, Sara T. Al‐Rashood, Faizah A. Binjubair, Marwa Alsulaimany, Hazem A. Ghabbour, Wagdy M. Eldehna, Hatem A. Abdel‐Aziz
Topics & Concepts
PyrazoleIn vivoSulfonamideCyclooxygenaseChemistryEnzymePharmacologyBiochemistryCombinatorial chemistryStereochemistryMedicineBiologyBiotechnologyInflammatory mediators and NSAID effectsSynthesis and biological activityComputational Drug Discovery Methods