Development of direct compression Acetazolamide tablet with improved bioavailability in healthy human volunteers enabled by cocrystallization with p-Aminobenzoic acid
Nimmy Kumari, Parag Roy, Sukanta Roy, Chenguang Wang, Sourav Das, Noopur Pandey, Susanta Mondal, Anirbandeep Bose, Changquan Calvin Sun, Animesh Ghosh
Topics & Concepts
CocrystalAcetazolamideBioavailabilityChemistryActive ingredientDosage formPharmacologyBiopharmaceuticalValdecoxibChromatographyMedicineOrganic chemistryAnesthesiaBiotechnologyMoleculeEnzymeBiologyHydrogen bondRofecoxibCyclooxygenaseCrystallography and molecular interactionsCrystallization and Solubility StudiesEnergetic Materials and Combustion