Synthesis and evaluation of novel arylisoxazoles linked to tacrine moiety: in vitro and in vivo biological activities against Alzheimer’s disease
Arezoo Rastegari, Maliheh Safavi, Fahimeh Vafadarnejad, Zahra Najafi, Roshanak Hariri, Syed Nasir Abbas Bukhari, Aida Iraji, Najmeh Edraki, Omidreza Firuzi, Mina Saeedi, Mohammad Mahdavi, Tahmineh Akbarzadeh
Topics & Concepts
TacrineAcetylcholinesteraseButyrylcholinesteraseCholinesteraseIn vivoChemistryPharmacologyAchéIC50In vitroBiochemistryEnzymeMedicineBiologyBiotechnologyCholinesterase and Neurodegenerative DiseasesComputational Drug Discovery MethodsAlzheimer's disease research and treatments