A chemoinformatics search for peroxisome proliferator-activated receptors ligands revealed a new pan-agonist able to reduce lipid accumulation and improve insulin sensitivity
Sabina Sblano, Carmen Cerchia, Antonio Laghezza, Luca Piemontese, Leonardo Brunetti, Rosalba Leuci, Federica Gilardi, Aurélien Thomas, Massimo Genovese, Alice Santi, Paolo Tortorella, Paolo Paoli, Antonio Lavecchia, Fulvio Loiodice
Topics & Concepts
CheminformaticsChemistryPeroxisome proliferator-activated receptorReceptorAgonistPPAR agonistPeroxisomePharmacologyGlucose homeostasisNuclear receptorInsulin resistancePeroxisome proliferator-activated receptor gammaTroglitazoneInsulin sensitivityBiochemistryInsulinEndocrinologyBiologyTranscription factorGeneComputational chemistryPeroxisome Proliferator-Activated ReceptorsMetabolism, Diabetes, and CancerCancer, Lipids, and Metabolism